One-Pot Synthesis of Enantiopure Pyrrolopiperazines

Pertejo Fernández, Pablo; González Saiz, Beatriz; Quesada Pato, Roberto; García Valverde, María

doi:10.1021/acs.joc.0c02103

dc.contributor.author	Pertejo Fernández, Pablo
dc.contributor.author	González Saiz, Beatriz
dc.contributor.author	Quesada Pato, Roberto
dc.contributor.author	García Valverde, María
dc.date.accessioned	2021-03-16T09:06:09Z
dc.date.available	2021-03-16T09:06:09Z
dc.date.issued	2020-11
dc.identifier.issn	0022-3263
dc.identifier.uri	http://hdl.handle.net/10259/5648
dc.description.abstract	A simple one-pot protocol for the synthesis of fused pyrrolopiperazines with a complete diastereoselectivity has been developed. This novel methodology combined the Ugi reaction with a spontaneous enamine alkylation on a multicomponent domino reaction, starting from nonprotected diamines and arylglyoxals.	en
dc.description.sponsorship	Consejerıá de Educacioń de la Junta de Castilla y León (project BU075G19)	es
dc.format.mimetype	application/pdf
dc.language.iso	eng	es
dc.publisher	American Chemical Society	es
dc.relation.ispartof	The Journal of Organic Chemistry. 2020, V. 85, n. 21, p. 14240–14245	es
dc.subject.other	Química orgánica	es
dc.subject.other	Chemistry, Organic	en
dc.title	One-Pot Synthesis of Enantiopure Pyrrolopiperazines	en
dc.type	info:eu-repo/semantics/article
dc.rights.accessRights	info:eu-repo/semantics/openAccess
dc.relation.publisherversion	https://doi.org/10.1021/acs.joc.0c02103
dc.identifier.doi	10.1021/acs.joc.0c02103
dc.relation.projectID	info:eu-repo/grantAgreement/JCyL/BU075G19
dc.identifier.essn	1520-6904
dc.journal.title	The Journal of Organic Chemistry	es
dc.volume.number	85	es
dc.issue.number	21	es
dc.page.initial	14240	es
dc.page.final	14245	es
dc.type.hasVersion	info:eu-repo/semantics/acceptedVersion

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